Structure/Class |
- Phencyclidine derivative
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Pharmacodynamics |
- NMDA receptor antagonist. It is the only IV anaesthetic agent that has significant analgesic properties
- Organ system effects as follows:
- CNS
- It is a cerebral vasodilator and tends to increase cerebral blood flow and cerebral metabolic rate. Therefore, it is contra-indicated in RICP.
- May be used for status epilepticus if other means are unsuccessful.
- Emergence phenomenon – tends to be less severe and of lower incidence in children. Premedication with BZD may decrease incidence.
- CVS
- It produces transient by significant centrally mediated stimulation, therefore increasing HR and cardiac output.
- It is thought to be a direct myocardial depressant, and this property may become apparent in the patients that are critically ill and have limited ability to increase their sympathetic drive.
- Respiratory
- Transient apnoea and hypoventilation if large dose given rapidly.
- Importantly – causes lacrimation and salivation. May cause laryngospasm in children.
- Relaxes bronchial s/m: consider in severe asthma
- If used as a single drug, the respiratory response to hypoxia and hypercapnia is NOT affected
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Absorption/administration |
- IV or IM.
- Can be given as bolus/infusion
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Distribution |
- Very lipid soluble
- Only IV anaesthetic agent that has low protein binding
- Large Vd – 3L/kg
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Metabolism |
- Metabolised in the liver to norketamine (an active metabolite) and then conjugated to water soluble metabolites and excreted in the urine.
- Distribution T ½: 11-16 minutes
- Elimination T ½ : 2-4 hours
- Duration of action: 5-10 minutes
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Excretion |
- Urine
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Indications |
- Procedural sedation (Very useful in children – give IM)
- Intravenous anaesthetic for induction
- Pain management
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Contraindications |
- Head injury and RICP are absolute CI.
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Special precautions |
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Interactions |
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Adverse events |
- Salivation/bronchorrhoea, leading to laryngospasm
- Emergence phenomena
- RICP
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Dosing/administration |
- 1-2mg/kg if induction
- Pain dose is 0.1mg/kg, infusion is 0.1mg-0.3mg/kg
- 4mg/kg IM if procedural sedation
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Toxicology |
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Withdrawal syndrome |
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Special notes |
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